Detalhe da pesquisa
1.
Clinical targeting of HIV capsid protein with a long-acting small molecule.
Nature
; 584(7822): 614-618, 2020 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-32612233
2.
Lenacapavir: A Novel, Potent, and Selective First-in-Class Inhibitor of HIV-1 Capsid Function Exhibits Optimal Pharmacokinetic Properties for a Long-Acting Injectable Antiretroviral Agent.
Mol Pharm
; 20(12): 6213-6225, 2023 Dec 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-37917742
3.
A highly potent long-acting small-molecule HIV-1 capsid inhibitor with efficacy in a humanized mouse model.
Nat Med
; 25(9): 1377-1384, 2019 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-31501601
4.
Sequence-selective DNA recognition: natural products and nature's lessons.
Chem Biol
; 11(12): 1607-17, 2004 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-15610844
5.
A fluorescent intercalator displacement assay for establishing DNA binding selectivity and affinity.
Curr Protoc Nucleic Acid Chem
; Chapter 8: Unit 8.5, 2005 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-18428943
6.
A fluorescent intercalator displacement assay for establishing DNA binding selectivity and affinity.
Acc Chem Res
; 37(1): 61-9, 2004 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-14730995
7.
Comprehensive high-resolution analysis of hairpin polyamides utilizing a fluorescent intercalator displacement (FID) assay.
Bioorg Med Chem
; 11(20): 4479-86, 2003 Oct 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-13129584
8.
High-resolution assessment of protein DNA binding affinity and selectivity utilizing a fluorescent intercalator displacement (FID) assay.
Bioorg Med Chem Lett
; 13(21): 3805-7, 2003 Nov 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-14552784
9.
Determination of binding affinities of triplex forming oligonucleotides using a fluorescent intercalator displacement (FID) assay.
Bioorg Med Chem Lett
; 13(21): 3801-4, 2003 Nov 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-14552783